Modulating Pharmacokinetics, Tumor Uptake and Biodistribution by Engineered Nanoparticles Nanoparticle Surface Charge and Biodistribution
2011

How Nanoparticle Surface Charge Affects Tumor Uptake

Sample size: 3 publication 10 minutes Evidence: moderate

Author Information

Author(s): Arvizo Rochelle R., Miranda Oscar R., Moyano Daniel F., Walden Chad A., Giri Karuna, Bhattacharya Resham, Robertson J. David, Rotello Vincent M., Reid Joel M., Mukherjee Priyabrata

Primary Institution: Mayo Clinic Rochester

Hypothesis

The neutral and zwitterionic nanoconjugates would exhibit increased tumor uptake relative to negative and positively charged analogs.

Conclusion

Neutral and zwitterionic nanoparticles demonstrated longer circulation time and enhanced tumor uptake compared to negatively and positively charged nanoparticles.

Supporting Evidence

  • Neutral and zwitterionic nanoparticles had longer circulation times.
  • Negatively and positively charged nanoparticles had shorter half-lives.
  • Tumor uptake was enhanced by neutral and zwitterionic nanoparticles.
  • The study used a family of structurally homologous nanoparticles.

Takeaway

Some tiny particles can help medicine get to the right place in the body better than others, depending on how they are made.

Methodology

The study involved injecting different types of nanoparticles into mice and measuring their circulation time and tumor uptake.

Limitations

The study primarily focused on a specific type of nanoparticle and may not generalize to all nanoparticles.

Participant Demographics

Male CD1 mice and athymic nude mice were used in the experiments.

Digital Object Identifier (DOI)

10.1371/journal.pone.0024374

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