Haloperidol treatment induces tissue- and sex-specific changes in DNA methylation: a control study using rats
2006

Haloperidol Treatment and DNA Methylation Changes in Rats

Sample size: 40 publication Evidence: moderate

Author Information

Author(s): Shimabukuro Morihiro, Jinno Yoshihiro, Fuke Chiaki, Okazaki Yuji

Primary Institution: Ryukyu University School of Medicine

Hypothesis

Is the difference in global methylation state of blood leukocyte DNA between male subjects with and without schizophrenia a primary effect of the disease state or a secondary effect of antipsychotics?

Conclusion

Haloperidol affects DNA methylation states in the brain and other tissues, suggesting a role for antipsychotic drugs in the observed disparity in methylation content in male subjects with schizophrenia.

Supporting Evidence

  • Haloperidol treatment decreased mC content in male rat leukocytes.
  • Haloperidol treatment increased mC content in female rat leukocytes.
  • Significant decrease in mC content in the brain of female rats treated with haloperidol.
  • Haloperidol treatment resulted in increased mC content in the liver for both sexes.

Takeaway

This study looked at how a drug called haloperidol changes DNA in rats, finding that it affects how DNA is marked in different ways for male and female rats.

Methodology

Rats were given daily injections of haloperidol or a placebo for 21 days, and their DNA methylation was analyzed using high performance liquid chromatography.

Potential Biases

Potential bias due to the limited sample size and the specific model used (rats) which may not fully represent human conditions.

Limitations

The study used a limited number of rats and could not demonstrate a causative effect of haloperidol on hypomethylation in male patients with schizophrenia.

Participant Demographics

40 male and female Sprague-Dawley rats.

Statistical Information

P-Value

0.026

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1186/1744-9081-2-37

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