Development and Characterization of Novel Combinations and Compositions of Nanostructured Lipid Carrier Formulations Loaded with Trans-Resveratrol for Pulmonary Drug Delivery
2024

Nanostructured Lipid Carrier Formulations for Pulmonary Drug Delivery

publication 10 minutes Evidence: high

Author Information

Author(s): Khan Iftikhar, Sunita, Hussein Nozad R., Omer Huner K., Elhissi Abdelbary, Houacine Chahinez, Khan Wasiq, Yousaf Sakib, Rathore Hassaan A., Fernández García Raquel, Bolás-Fernández Francisco, Fraguas-Sánchez Ana Isabel

Primary Institution: School of Pharmacy and Biomolecular Sciences, Liverpool John Moores University

Hypothesis

This study aimed to fabricate, optimize, and characterize nanostructured lipid carriers (NLCs) loaded with trans-resveratrol (TRES) for pulmonary drug delivery.

Conclusion

Formulation F14, combined with an air-jet nebulizer, demonstrated superior stability and aerosolization performance for pulmonary drug delivery.

Supporting Evidence

  • Formulation F14 showed greater stability at 4 and 25 °C for six months.
  • F14 exhibited higher emitted dose (ED; 80%) and fine particle dose (FPD; 1150 µg).
  • The study demonstrated that TRES-NLC formulations can effectively target the pulmonary system.

Takeaway

Researchers created a special type of tiny fat particles to deliver a medicine called trans-resveratrol to the lungs, and they found one version worked best.

Methodology

The study involved preparing 24 different formulations of TRES-NLCs using hot, high-pressure homogenization and evaluating their physicochemical properties and stability.

Limitations

The study did not specify participant demographics or clinical trials, focusing instead on laboratory formulations.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.3390/pharmaceutics16121589

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