Plasmodium falciparum glutamate dehydrogenase a is dispensable and not a drug target during erythrocytic development
2011

The Role of Plasmodium falciparum Glutamate Dehydrogenase A in Parasite Development

publication 10 minutes Evidence: moderate

Author Information

Author(s): Janet Storm, Jan Perner, Isabela Aparicio, Eva-Maria Patzewitz, Kellen Olszewski, Manuel Llinas, Paul C Engel, Sylke Müller

Primary Institution: University of Glasgow

Hypothesis

Is GDHa a suitable drug target during the intra-erythrocytic development of Plasmodium falciparum?

Conclusion

GDHa is not essential for the growth of Plasmodium falciparum and is unlikely to be a suitable target for drug development.

Supporting Evidence

  • The absence of GDHa did not affect the growth of the mutant parasites under low or elevated oxygen conditions.
  • GDHa null mutants showed no significant changes in the expression of antioxidant proteins.
  • Metabolic labeling experiments indicated that GDHa is not essential for the conversion of glutamate to α-ketoglutarate.

Takeaway

The malaria parasite can grow just fine without a specific enzyme called GDHa, which means it might not be a good target for new medicines.

Methodology

The study involved creating GDHa null mutants of P. falciparum and assessing their growth and metabolic functions under various conditions.

Limitations

The study was conducted under in vitro conditions, which may not fully represent the in vivo environment of the parasite.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1186/1475-2875-10-193

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