1,2-Dithiol-3-thione and dithioester analogues: potential radioprotectors
1990

Potential Radioprotectors from Dithiol Compounds

publication Evidence: moderate

Author Information

Author(s): B.A. Teicher, J. Stemwedel, T.S. Herman, P.K. Ghoshal, A. Rosowsky

Primary Institution: Dana-Farber Cancer Institute

Hypothesis

Can 1,2-dithiol-3-thione and dithioester compounds act as effective radioprotectors in EMT6 cells?

Conclusion

Several 1,2-dithiol-3-thione and dithioester compounds were found to be effective radioprotectors in vitro.

Supporting Evidence

  • 1,2-dithiol-3-thiones were generally more cytotoxic than dithioesters.
  • The 5-(2-thienyl)-1,2-dithiol-3-thione produced a radiation protection factor of 2.7.
  • Several dithioesters showed radiation protection factors ranging from 2.6 to 2.9.

Takeaway

Some special chemicals can help protect cells from radiation damage, which is important for cancer treatment.

Methodology

The study tested various 1,2-dithiol-3-thione and dithioester compounds for their radioprotective effects on EMT6 cells in vitro.

Limitations

The study was conducted in vitro, and the effects in vivo are still being investigated.

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