tert-Butyl N-((1S)-2-hy­droxy-1-{N′-[(1E)-4-meth­oxy­benzyl­idene]hydrazinecarbon­yl}eth­yl)carbamate
2011

Study of a New Compound for Anti-Tumor Activity

publication Evidence: moderate

Author Information

Author(s): Alessandra C. Pinheiro, Marcus V. N. de Souza, Edward R. T. Tiekink, Solange M. S. V. Wardell, James L. Wardell

Primary Institution: Fundação Oswaldo Cruz, Instituto de Tecnologia, em Fármacos – Farmanguinhos

Hypothesis

The study investigates the structural properties of a new compound derived from L-serine and its potential anti-tumor activity.

Conclusion

The compound exhibits a unique molecular structure with significant hydrogen bonding interactions that may contribute to its biological activity.

Supporting Evidence

  • The compound's structure was characterized by a dihedral angle of 79.6° between amide residues.
  • Hydrogen bonding interactions were observed between hydroxy, amine, and carbonyl groups.
  • The synthesis yielded only the E isomer after recrystallization.

Takeaway

Scientists created a new molecule that might help fight cancer, and they found that its structure is really interesting because of how its parts stick together.

Methodology

The compound was synthesized from L-serine and 4-methoxybenzaldehyde, followed by crystallization and structural analysis using X-ray diffraction.

Limitations

The absolute structure of the compound could not be determined experimentally.

Digital Object Identifier (DOI)

10.1107/S1600536811024263

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