Bioequivalence study of three ibuprofen formulations after single dose administration in healthy volunteers
2008

Bioequivalence Study of Eudorlin® Extra and Two Reference Ibuprofen Formulations

Sample size: 60 publication 10 minutes Evidence: moderate

Author Information

Author(s): Bramlage Peter, Goldis Adrian

Primary Institution: Institute for Clinical Pharmacology, Medical Faculty Carl Gustav Carus, Technical University Dresden

Hypothesis

The study aims to determine the bioavailability and bioequivalence of Eudorlin® extra compared to Nurofen® forte and Migränin® after single dose administration.

Conclusion

Eudorlin® extra is bioequivalent to Nurofen® forte and Migränin® in terms of absorption rate and extent, but reaches higher peak plasma concentrations more quickly.

Supporting Evidence

  • Eudorlin® extra showed a higher Cmax compared to both reference products.
  • The time to maximum plasma concentration (tmax) was shorter for Eudorlin® extra.
  • All pharmacokinetic parameters were within the acceptance range set by EMEA.

Takeaway

This study shows that a new ibuprofen product works just as well as two other brands, but it gets into your system faster and stronger.

Methodology

A randomized, open label, multiple sequence cross-over study with a wash-out period of 7–10 days was conducted.

Potential Biases

There may be a risk of bias due to the open-label design.

Limitations

The study had a small sample size and only included healthy volunteers.

Participant Demographics

60 healthy volunteers, 41 male and 19 female, aged 20 to 45 years.

Statistical Information

P-Value

0.0014

Confidence Interval

90% CI for AUC0-t(last) and AUC0-∞ within 80-125%; Cmax within 75-133%

Statistical Significance

p<0.0001

Digital Object Identifier (DOI)

10.1186/1471-2210-8-18

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