Polyene Macrolide Antifungal Drugs Trigger Interleukin-1β Secretion by Activating the NLRP3 Inflammasome
2011

Polyene Macrolide Antifungal Drugs Trigger IL-1β Secretion

Sample size: 3 publication Evidence: high

Author Information

Author(s): Darisipudi Murthy Narayana, Allam Ramanjaneyulu, Rupanagudi Khader Valli, Anders Hans-Joachim

Primary Institution: Medizinische Poliklinik, University of Munich, Munich, Germany

Hypothesis

Do polyene macrolide antifungal drugs activate the NLRP3 inflammasome to induce IL-1β secretion?

Conclusion

Polyene macrolide antifungal drugs activate the NLRP3 inflammasome and induce IL-1β secretion in dendritic cells.

Supporting Evidence

  • Amphotericin B, nystatin, and natamycin induce high levels of IL-1β secretion in dendritic cells.
  • IL-1β secretion requires both the induction of pro-IL-1β and activation of caspase-1.
  • NLRP3 is essential for drug-induced IL-1β release.
  • Potassium efflux is a necessary step for NLRP3 activation by these antifungal drugs.

Takeaway

Some antifungal drugs can help our body's immune system fight infections by making it release a special chemical called IL-1β.

Methodology

The study involved exposing LPS-primed bone marrow-derived dendritic cells to antifungal drugs and measuring IL-1β production in cell culture supernatants.

Participant Demographics

C57BL/6 mouse bone marrow-derived dendritic cells and macrophages were used.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0019588

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