Preclinical evaluation of the antineoplastic action of 5-aza-2'-deoxycytidine and different histone deacetylase inhibitors on human Ewing's sarcoma cells
2008

Combining 5AZA-CdR and HDAC Inhibitors for Ewing's Sarcoma Treatment

publication Evidence: moderate

Author Information

Author(s): Annie Hurtubise, Mark L Bernstein, Richard L Momparler

Primary Institution: Département de pharmacologie, Université de Montréal

Hypothesis

Does the combination of 5-aza-2'-deoxycytidine and histone deacetylase inhibitors enhance antineoplastic activity against Ewing's sarcoma cells?

Conclusion

The combination of 5AZA-CdR and MS-275 shows significant potential for treating advanced Ewing's sarcoma by reactivating tumor suppressor genes.

Supporting Evidence

  • 5AZA-CdR reactivates silenced tumor suppressor genes.
  • HDAC inhibitors enhance the antineoplastic action of 5AZA-CdR.
  • The combination of 5AZA-CdR and MS-275 showed marked synergy.
  • The study suggests further clinical investigation of this combination.

Takeaway

This study found that using two types of cancer-fighting drugs together can work better than using them alone to help treat a specific type of cancer called Ewing's sarcoma.

Methodology

The study used clonogenic assays to evaluate the antineoplastic activity of 5AZA-CdR combined with various HDAC inhibitors on Ewing's sarcoma cell lines.

Statistical Information

P-Value

p < 0.01

Statistical Significance

p < 0.01

Digital Object Identifier (DOI)

10.1186/1475-2867-8-16

Want to read the original?

Access the complete publication on the publisher's website

View Original Publication