Will histone deacetylase inhibitors require combination with other agents to fulfil their therapeutic potential?
2008

Combining Histone Deacetylase Inhibitors with Other Cancer Treatments

publication Evidence: moderate

Author Information

Author(s): Nolan L, Johnson P W M, Ganesan A, Packham G, Crabb S J

Primary Institution: Cancer Research UK Clinical Centre, School of Medicine, University of Southampton

Hypothesis

In most scenarios, combination with other therapeutic modalities will be required to optimise efficacy of histone deacetylase inhibitors.

Conclusion

Histone deacetylase inhibitors show promise when combined with various anticancer agents, potentially enhancing their effectiveness.

Supporting Evidence

  • Histone deacetylase inhibitors have shown modest antitumor activity in initial clinical trials.
  • Combination with cytotoxic chemotherapy has demonstrated synergistic effects in pre-clinical models.
  • Clinical trials are ongoing to evaluate the effectiveness of HDI combinations with various agents.

Takeaway

Histone deacetylase inhibitors are like helpers for cancer treatments, making them work better when used together.

Methodology

This review discusses the mechanisms and evidence supporting the combination of HDAC inhibitors with other cancer therapies.

Limitations

The study primarily relies on pre-clinical data and early-phase clinical trials, limiting the generalizability of findings.

Digital Object Identifier (DOI)

10.1038/sj.bjc.6604557

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