Specifically blocking αvβ8-mediated TGF-β signaling to reverse immunosuppression by modulating macrophage polarization
2025

Blocking αvβ8 to Reverse Immunosuppression in Tumors

Sample size: 10 publication 10 minutes Evidence: high

Author Information

Author(s): Guo Cuicui, Sun Hui, Du Yulei, Dai Xiaodong, Pang Yu, Han Zhen, Xiong Xinhui, Li Shaowei, Zhang Junhua, Zheng Qingbing, Gui Xun

Primary Institution: Mabwell (Shanghai) Bioscience Co., Ltd, Shanghai, China

Hypothesis

Can blocking αvβ8-mediated TGF-β signaling enhance anti-tumor immunity?

Conclusion

Targeting αvβ8 with a blocking antibody significantly inhibits tumor growth by enhancing immune cell infiltration and modulating macrophage polarization.

Supporting Evidence

  • Integrin αvβ8 is expressed in certain tumor types and tumor-infiltrating macrophages.
  • The specific αvβ8 antibody 130H2 demonstrated high affinity and blocking potency.
  • Combining the antibody with PD-1 inhibition produced a synergistic anti-tumor effect.
  • Blocking αvβ8 significantly increased immune cell infiltration in tumors.
  • Pharmacokinetic studies showed favorable properties in cynomolgus monkeys.

Takeaway

This study shows that a special antibody can help the immune system fight tumors better by changing how certain immune cells work.

Methodology

Single-cell RNA sequencing was used to analyze αvβ8 expression, and an anti-αvβ8 antibody was developed and tested in vitro and in mouse models.

Participant Demographics

Ten male patients aged 50 to 75 with kidney renal clear cell carcinoma.

Statistical Information

P-Value

p<0.01

Statistical Significance

p<0.01

Digital Object Identifier (DOI)

10.1186/s13046-024-03250-1

Want to read the original?

Access the complete publication on the publisher's website

View Original Publication