Different pH requirements are associated with divergent inhibitory effects of chloroquine on human and avian influenza A viruses
2007

Chloroquine's Effects on Human and Avian Influenza A Viruses

publication Evidence: moderate

Author Information

Author(s): Di Trani Livia, Savarino Andrea, Campitelli Laura, Norelli Sandro, Puzelli Simona, D'Ostilio Daniela, Vignolo Edoardo, Donatelli Isabella, Cassone Antonio

Primary Institution: Istituto Superiore di Sanità, Rome, Italy

Hypothesis

Does the low pH-dependency of influenza A viruses affect the antiviral effects of chloroquine?

Conclusion

Chloroquine inhibits the replication of influenza A viruses that require low pH for proper fusion activation.

Supporting Evidence

  • Chloroquine showed a dose-dependent inhibition of the H5N9 virus with an EC50 of 14.38 μM.
  • The inhibitory effect of chloroquine was maximal when added at the time of infection.
  • A correlation was found between the electrostatic potential of the HA2 subunit and the EC50 of chloroquine.

Takeaway

Chloroquine can help stop certain flu viruses from spreading by working best when the virus is trying to enter cells, especially when the environment is acidic.

Methodology

The study tested chloroquine's antiviral effects on various human and avian influenza A viruses using cell cultures and measured viral replication.

Limitations

The study primarily focused on in vitro conditions, which may not fully represent in vivo responses.

Statistical Information

P-Value

0.024

Statistical Significance

p = 0.024

Digital Object Identifier (DOI)

10.1186/1743-422X-4-39

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