Antiviral Activity of 3(2H)- and 6-Chloro-3(2H)-Isoflavenes against Highly Diverged, Neurovirulent Vaccine-Derived, Type2 Poliovirus Sewage Isolates
2011

Antiviral Activity of Isoflavenes Against Vaccine-Derived Poliovirus

Sample size: 10 publication 10 minutes Evidence: moderate

Author Information

Author(s): Shulman Lester M., Sofer Danit, Manor Yossi, Mendelson Ella, Balanant Jean, Salvati Anna Laura, Delpeyroux Francis, Fiore Lucia

Primary Institution: Central Virology Laboratory, Public Health Services Israel Ministry of Health

Hypothesis

Do highly evolved vaccine-derived polioviruses retain sensitivity to isoflavenes?

Conclusion

Isoflavenes effectively reduced viral loads in vitro against most highly-diverged vaccine-derived polioviruses.

Supporting Evidence

  • Isoflavenes inhibited viral titers of Sabin-2 and nine of ten aVDPV2s by one to two log10.
  • The tenth aVDPV2 isolate was unaffected by both isoflavenes.
  • All aVDPV2 isolates reverted to a neurovirulent phenotype except one with specific amino acid substitutions.

Takeaway

Researchers tested two compounds to see if they could stop a type of poliovirus from growing, and they found that most of the viruses were still affected by the compounds.

Methodology

The study involved titering poliovirus isolates on HEp2C cells in the presence of isoflavenes and assessing neurovirulence in transgenic mice.

Limitations

The study did not evaluate the in vivo effectiveness of isoflavenes in humans.

Statistical Information

P-Value

p<0.01

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0018360

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