High-dose tamoxifen as an enhancer of etoposide cytotoxicity. Clinical effects and in vitro assessment in p-glycoprotein expressing cell lines
1992

High-dose tamoxifen enhances etoposide effectiveness in cancer treatment

Sample size: 26 publication Evidence: moderate

Author Information

Author(s): N.S.A. Stuart, P. Philip, A.L. Harris, K. Tonkin, S. Houlbrook, J. Kirk, E.A. Lien, J. Carmichael

Primary Institution: ICRF Clinical Oncology Unit, Churchill Hospital, Oxford

Hypothesis

Can high-dose tamoxifen enhance the cytotoxicity of etoposide in patients with drug-resistant cancer?

Conclusion

High-dose tamoxifen can be administered with acceptable toxicity but does not significantly enhance etoposide cytotoxicity in vitro.

Supporting Evidence

  • Two patients showed a partial response to the treatment.
  • Significant nausea was reported in a portion of the patients.
  • Serum levels of tamoxifen were sufficient to modulate drug resistance in vitro.

Takeaway

Doctors tested a combination of high-dose tamoxifen and etoposide on cancer patients, but it didn't work as well as hoped.

Methodology

Patients with relapsed or drug-resistant cancer were treated with oral etoposide and high-dose oral tamoxifen, followed by assessments of serum levels and toxicity.

Potential Biases

Potential bias due to lack of a control group and the subjective nature of reported symptoms.

Limitations

The study was small and primarily focused on safety rather than efficacy.

Participant Demographics

Median age was 50, with a mix of male and female patients and various cancer types.

Statistical Information

P-Value

p<0.01

Statistical Significance

p<0.05

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