Membrane androgen receptor activation triggers down-regulation of PI-3K/Akt/NF-kappaB activity and induces apoptotic responses via Bad, FasL and caspase-3 in DU145 prostate cancer cells
2008

Testosterone Triggers Apoptosis in Prostate Cancer Cells

publication Evidence: moderate

Author Information

Author(s): Papadopoulou Natalia, Charalampopoulos Ioannis, Anagnostopoulou Vasileia, Konstantinidis Georgios, Föller Michael, Gravanis Achilleas, Alevizopoulos Konstantinos, Lang Florian, Stournaras Christos

Primary Institution: Department of Biochemistry, University of Crete Medical School, Heraklion, Greece

Hypothesis

Membrane androgen receptors induce apoptosis in DU145 prostate cancer cells through specific signaling pathways.

Conclusion

Testosterone-albumin conjugates activate specific pro-apoptotic pathways in DU145 prostate cancer cells, suggesting their potential as anti-tumor agents.

Supporting Evidence

  • Testosterone-albumin conjugates down-regulated pro-survival pathways in DU145 cells.
  • FasL expression was significantly increased following treatment with testosterone-albumin.
  • Caspase-3 activity was activated in DU145 cells treated with testosterone-albumin.
  • PI-3K and Akt activities were suppressed after testosterone-albumin treatment.
  • Actin cytoskeleton disruption inhibited the apoptotic effects of testosterone-albumin.

Takeaway

When prostate cancer cells are treated with a special form of testosterone, they start to die because of changes inside the cells.

Methodology

The study involved treating DU145 prostate cancer cells with testosterone-albumin conjugates and measuring various apoptotic markers and signaling pathways.

Limitations

The study primarily focuses on one cell line and may not represent all prostate cancer types.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1186/1476-4598-7-88

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