The ETS Family Member TEL Binds to Nuclear Receptors RAR and RXR and Represses Gene Activation
2011

TEL Represses Gene Activation by Binding to RAR and RXR

publication Evidence: moderate

Author Information

Author(s): Magda A. Meester-Smoor, Marjolein J. F. W. ter Haar, W. Martijn van Wely, Karel H. M. Aarnoudse, Albert-Jan L. H. J. van Oord, Gertine van Tilburg, Gabrielle B. A. Zwarthoff, Ellen C. Z. van der Plas

Primary Institution: Erasmus MC, Rotterdam, The Netherlands

Hypothesis

TEL acts as a transcriptional repressor of RAR signaling by binding to RAR and RXR.

Conclusion

TEL is identified as a co-repressor of RAR-RXR-mediated transcription, functioning independently of histone deacetylases.

Supporting Evidence

  • TEL binds directly to RARα and RXRα, indicating its role in transcriptional repression.
  • The shorter isoform of TEL is a more efficient repressor of RAR signaling compared to the longer isoform.
  • Repression by TEL does not involve recruitment of histone deacetylases, suggesting alternative mechanisms.
  • Both HLH and DBD domains of TEL are crucial for its binding to RARα.

Takeaway

TEL is a protein that helps turn off certain genes by sticking to other proteins called RAR and RXR, which are important for cell growth and development.

Methodology

The study involved binding assays, transfection experiments in Hep3B cells, and luciferase reporter assays to assess transcriptional activity.

Limitations

The study does not explore the full range of biological processes influenced by TEL and RAR signaling.

Digital Object Identifier (DOI)

10.1371/journal.pone.0023620

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