Calbindin 2 (CALB2) Regulates 5-Fluorouracil Sensitivity in Colorectal Cancer by Modulating the Intrinsic Apoptotic Pathway
2011

CALB2 and Colorectal Cancer: How CALB2 Affects 5-FU Sensitivity

publication Evidence: moderate

Author Information

Author(s): Leanne Stevenson, Wendy L. Allen, Irina Proutski, Gail Stewart, Louise Johnston, Karen McCloskey, Peter M. Wilson, Daniel B. Longley, Patrick G. Johnston

Primary Institution: Queen's University Belfast, Belfast, Northern Ireland

Hypothesis

The study investigates the role of Calbindin 2 (CALB2) in regulating the response of colorectal cancer (CRC) cells to 5-Fluorouracil (5-FU).

Conclusion

CALB2 is involved in apoptosis induction through the intrinsic mitochondrial pathway, and its down-regulation may represent a mechanism of resistance to 5-FU in colorectal cancer cells.

Supporting Evidence

  • CALB2 expression was down-regulated in CRC cell lines following 5-FU treatment.
  • 5-FU-induced apoptosis was significantly reduced in CALB2-silenced CRC cell lines.
  • CALB2 translocated to the mitochondria following 5-FU treatment.
  • Co-silencing of XIAP overcame 5-FU resistance in CALB2-silenced cells.
  • The study identified pathways associated with 5-FU resistance, including calcium signaling and apoptosis.

Takeaway

CALB2 helps cancer cells die when treated with a drug called 5-FU, and if CALB2 is turned off, the cancer cells can survive the treatment better.

Methodology

The study used real-time RT-PCR, Western blot analysis, and flow cytometry to assess CALB2 expression and apoptosis in CRC cell lines treated with 5-FU.

Limitations

The study primarily focuses on in vitro models, which may not fully replicate the complexity of human tumors.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0020276

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