HOXC11–SRC-1 regulation of S100beta in cutaneous melanoma: new targets for the kinase inhibitor dasatinib
2011

Regulation of S100beta in Melanoma by HOXC11 and SRC-1

Sample size: 80 publication Evidence: moderate

Author Information

Author(s): deBlacam C, Byrne C, Hughes E, McIlroy M, Bane F, Hill A D K, Young L S

Primary Institution: Royal College of Surgeons in Ireland

Hypothesis

The study investigates the regulation of S100beta in cutaneous melanoma by HOXC11 and SRC-1 and the potential modulation by dasatinib.

Conclusion

The study defines a signaling mechanism regulating S100beta in melanoma, which can be modulated by dasatinib.

Supporting Evidence

  • HOXC11 and SRC-1 were significantly elevated in malignant melanoma compared to benign nevi.
  • Dasatinib reduced S100beta expression and migration in melanoma cell lines.
  • HOXC11 recruitment to the S100beta promoter was confirmed in primary melanoma cells.

Takeaway

This study looks at how certain proteins help control a marker for melanoma, and a drug called dasatinib can change this process.

Methodology

The study used immunohistochemistry, immunofluorescence, western blot, qPCR, ChIP, and migration assays to investigate the regulation of S100beta.

Participant Demographics

Patients with malignant melanoma and benign nevi.

Statistical Information

P-Value

P<0.001 and P=0.017

Statistical Significance

p<0.001

Digital Object Identifier (DOI)

10.1038/bjc.2011.193

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