Bioactive Markers Based Pharmacokinetic Evaluation of Extracts of a Traditional Medicinal Plant, Piper sarmentosum
2011

Pharmacokinetic Evaluation of Piper sarmentosum Extracts

Sample size: 18 publication 10 minutes Evidence: moderate

Author Information

Author(s): Hussain Khalid, Ismail Zhari, Sadikun Amirin, Pazillah Ibrahim

Primary Institution: Universiti Sains Malaysia

Hypothesis

The study aimed to evaluate the pharmacokinetics of ethanol extract of Piper sarmentosum in rats.

Conclusion

Pellitorine and sarmentine have good oral bioavailability, while sarmentosine is not absorbed from the gastrointestinal tract.

Supporting Evidence

  • Pellitorine exhibited maximum plasma concentration of 34.77 ng/mL.
  • Sarmentine showed maximum plasma concentration of 191.50 ng/mL.
  • Sarmentosine exhibited zero oral bioavailability.
  • Pellitorine was distributed in multiple tissues including the liver and heart.
  • Sarmentine was found in the intestinal wall and heart.

Takeaway

This study looked at how well certain compounds from a plant called Piper sarmentosum are absorbed and used by the body.

Methodology

The study used Sprague-Dawley rats to evaluate absorption, distribution, and excretion of the plant extracts through HPLC analysis.

Limitations

The study was limited to a small sample size and focused only on specific markers.

Participant Demographics

Male Sprague-Dawley rats, weighing approximately 313 ± 17 g.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1093/ecam/nep143

Want to read the original?

Access the complete publication on the publisher's website

View Original Publication