Highly brominated anthracenes as precursors for the convenient synthesis of 2,9,10-trisubstituted anthracene derivatives
2008

Synthesis of Brominated Anthracene Derivatives

publication Evidence: high

Author Information

Author(s): Cakmak Osman, Aydogan Leyla, Berkil Kiymet, Gulcin Ilhami, Buyukgungor Orhan

Primary Institution: Gaziosmanpasa University

Hypothesis

Can highly brominated anthracenes be used as precursors for synthesizing 2,9,10-trisubstituted anthracene derivatives?

Conclusion

The study successfully demonstrates an efficient synthesis of hexabromide 3 and tribromide 12, which can be used to create various anthracene derivatives.

Supporting Evidence

  • The synthesis of hexabromide 3 was achieved in 95% yield without other stereoisomers.
  • Tribromide 12 was produced in 75% yield through a base-induced elimination reaction.
  • The methodology allows for the selective preparation of various anthracene derivatives.

Takeaway

The researchers found a new way to make special types of anthracene compounds using bromine without needing a catalyst.

Methodology

The study involved bromination of 9,10-dibromoanthracene and subsequent reactions to produce various anthracene derivatives.

Digital Object Identifier (DOI)

10.3762/bjoc.4.50

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